Bufadienolides from Kalanchoe daigremontiana as thrombin inhibitors— In vitro and in silico study

Author:

Kolodziejczyk-Czepas Joanna,Sieradzka Malgorzata,Moniuszko-Szajwaj Barbara,Pecio Łukasz,Ponczek Michal B.,Nowak Pawel,Stochmal Anna

Funder

National Science Centre

University of Lodz

Publisher

Elsevier BV

Subject

Molecular Biology,General Medicine,Biochemistry,Structural Biology

Reference35 articles.

1. Thrombin plasticity;Huntington;Biochim. Biophys. Acta,2012

2. Peptidomimetic thrombin inhibitors;Kikelj;Pathophysiol. Haemost. Thromb.,2003

3. Platelet glycoprotein Ib alpha binds to thrombin anion-binding exosite II inducing allosteric changes in the activity of thrombin;Li;J. Biol. Chem.,2001

4. Redesigning the monovalent cation specificity of an enzyme;Prasad;Proc. Natl. Acad. Sci. U. S. A.,2003

5. The miracle plant (Kalanchoe pinnata): a phytochemical and pharmacological review;Ahamad Aejazuddin;Int. J. Res. Ayurveda Pharm.,2011

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