Voltage-sensor conformation shapes the intra-membrane drug binding site that determines gambierol affinity in Kv channels
Author:
Funder
Vlaams Instituut voor de bevordering
Belgian Research Fund Flanders
FWO
IUAP
OT
Publisher
Elsevier BV
Subject
Cellular and Molecular Neuroscience,Pharmacology
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4. Block of voltage-gated potassium channels by Pacific ciguatoxin-1 contributes to increased neuronal excitability in rat sensory neurons;Birinyi-Strachan;Toxicol. Appl. Pharmacol.,2005
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4. Diastereoselective Ring-Closing Metathesis as a Means to Construct Medium-Sized Cyclic Ethers: Application to the Synthesis of a Photoactivatable Gambierol Derivative;The Journal of Organic Chemistry;2016-09-02
5. Gambierol and n-alkanols inhibit Shaker Kv channel via distinct binding sites outside the K+ pore;Toxicon;2016-09
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