(E)-1-(Heterocyclyl or cyclohexyl)-2-[1,3,7-trisubstituted (xanthin-8-yl)] ethenes as A2a adenosine receptor antagonists
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference29 articles.
1. Adenosine A1 and A2 receptors: Structure–function relationships
2. 8-Aryl- and 8-cycloalkyl-1,3-dipropylxanthines: further potent and selective antagonists for A1-adenosine receptors
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1. Synthesis of a New Series of 1H-Imidazol-1-yl Substituted 8-Phenylxanthines as Adenosine Receptor Ligands;Chemistry & Biodiversity;2011-07
2. Xanthines as Adenosine Receptor Antagonists;Methylxanthines;2010-08-19
3. ChemInform Abstract: (E)-1-(Heterocyclyl or Cyclohexyl)-2-(1,3,7-trisubstituted(xanthin-8- yl))ethenes as A2a Adenosine Receptor Antagonists.;ChemInform;2010-08-05
4. A2A Receptor Ligands: Past, Present and Future Trends;Current Topics in Medicinal Chemistry;2010-06-01
5. An efficient route to xanthine based A2A adenosine receptor antagonists and functional derivatives;Organic & Biomolecular Chemistry;2010
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