Inverse agonists at the polyamine-sensitive modulatory site of the NMDA receptor: 50-fold increase in potency by insertion of an aromatic ring into an alkanediamine chain-Reference-Cited by-同舟云学术

Inverse agonists at the polyamine-sensitive modulatory site of the NMDA receptor: 50-fold increase in potency by insertion of an aromatic ring into an alkanediamine chain

Published:1998-01 Issue:1 Volume:33 Page:3-14
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Berger Michael L.,Schödl Clemens,Noe Christian R.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference29 articles.

1. Modulation of the NMDA receptor by polyamines

2. Modulation of channel function by polyamines

3. Characterization of polyamines having agonist, antagonist, and inverse agonist effects at the polyamine recognition site of the NMDA receptor

4. Interaction of long chain n-alkyl diamines with the NMDA receptor complex

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