BCR-ABL1 Compound Mutations Combining Key Kinase Domain Positions Confer Clinical Resistance to Ponatinib in Ph Chromosome-Positive Leukemia

Author:

Zabriskie Matthew S.,Eide Christopher A.,Tantravahi Srinivas K.,Vellore Nadeem A.,Estrada Johanna,Nicolini Franck E.,Khoury Hanna J.,Larson Richard A.,Konopleva Marina,Cortes Jorge E.,Kantarjian Hagop,Jabbour Elias J.,Kornblau Steven M.,Lipton Jeffrey H.,Rea Delphine,Stenke Leif,Barbany Gisela,Lange Thoralf,Hernández-Boluda Juan-Carlos,Ossenkoppele Gert J.,Press Richard D.,Chuah Charles,Goldberg Stuart L.,Wetzler Meir,Mahon Francois-Xavier,Etienne Gabriel,Baccarani Michele,Soverini Simona,Rosti Gianantonio,Rousselot Philippe,Friedman Ran,Deininger Marie,Reynolds Kimberly R.,Heaton William L.,Eiring Anna M.,Pomicter Anthony D.,Khorashad Jamshid S.,Kelley Todd W.,Baron Riccardo,Druker Brian J.,Deininger Michael W.,O’Hare Thomas

Funder

Huntsman Cancer Institute

NIH

NCI

American Society of Hematology

Leukemia & Lymphoma Society

Howard Hughes Medical Institute

NCI MERIT award

Leukemia & Lymphoma Society (LLS) Scholar in Clinical Research

University of Utah Department of Medicinal Chemistry, a computing allocation at the XSEDE supercomputers

Office of Science of the U.S. Department of Energy

Publisher

Elsevier BV

Subject

Cancer Research,Cell Biology,Oncology

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