Molecular determinants of peptide and nonpeptide NK-2 receptor antagonists binding sites of the human tachykinin NK-2 receptor by site-directed mutagenesis-Reference-Cited by-同舟云学术

Molecular determinants of peptide and nonpeptide NK-2 receptor antagonists binding sites of the human tachykinin NK-2 receptor by site-directed mutagenesis

Published:2000-07 Issue:8 Volume:39 Page:1422-1429
ISSN:0028-3908
Container-title:Neuropharmacology
language:en
Short-container-title:Neuropharmacology

Author:

Giolitti Alessandro,Cucchi Paola,Renzetti Anna Rita,Rotondaro Luigi,Zappitelli Sabrina,Maggi Carlo Alberto

Publisher

Elsevier BV

Subject

Cellular and Molecular Neuroscience,Pharmacology

Reference27 articles.

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2. MEN 11420 (Nepadutant), a novel glycosylated bicyclic peptide tachykinin NK2 receptor antagonist;Catalioto;Br. J. Pharmacol.,1998

3. Conserved polar residues in the transmembrane domain of the human tachykinin NK2 receptor: functional roles and structural implications;Donnelly;Biochem. J.,1999

4. A potent and selective non-peptide antagonist of the neurokinin a (NK2) receptor

5. Mutational analysis of neurokinin receptor function;Fong;Can. J. Physiol. Pharmacol.,1995

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