Brain uptake and receptor binding of two [11C]labelled selective high affinity NK1-antagonists, GR203040 and GR205171 — PET studies in rhesus monkey-Reference-Cited by-同舟云学术

Brain uptake and receptor binding of two [11C]labelled selective high affinity NK1-antagonists, GR203040 and GR205171 — PET studies in rhesus monkey

Published:2000-03 Issue:4 Volume:39 Page:664-670
ISSN:0028-3908
Container-title:Neuropharmacology
language:en
Short-container-title:Neuropharmacology

Author:

Bergström M,Fasth K.-J,Kilpatrick G,Ward P,Cable K.M,Wipperman M.D,Sutherland D.R,Långström B

Publisher

Elsevier BV

Subject

Cellular and Molecular Neuroscience,Pharmacology

Reference14 articles.

1. The pharmacology of GR203040, a novel, potent and selective non-peptide tachykinin NK1 receptor antagonist;Beattie;British Journal of Pharmacology,1995

2. Measurement of human cerebral monoamine oxidase type B (MAO-B) activity with positron emission tomography (PET): a dose ranging study with the reversible inhibitor Ro 19-6327;Bench;European Journal of Clinical Pharmacology,1991

3. MAO-A inhibition in brain after dosing of Esuprone, Moclobemide and placebo in healthy volunteers — in vivo studies with positron emission tomography;Bergström;European Journal of Clinical Pharmacology,1997

4. In vitro and in vivo studies of substance P receptor expression in rats with the new analogue (Indium-111-DTPA-Arg)substance P;Breeman;Journal of Nuclear Medicine,1996

5. Synthesis of a nonpeptide carbon-11 labelled substance P antagonist for PET studies;Del-Rosario;Nuclear Medicine and Biology,1993

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