Shielding effects at 17α-substituted estrogens. A tentative explanation for the low biological activity of 17α-ethyl-estradiol based on I.R. and NMR spectroscopic studies-Reference-Cited by-同舟云学术

Shielding effects at 17α-substituted estrogens. A tentative explanation for the low biological activity of 17α-ethyl-estradiol based on I.R. and NMR spectroscopic studies

Published:1985-11 Issue:5 Volume:23 Page:611-616
ISSN:0022-4731
Container-title:Journal of Steroid Biochemistry
language:en
Short-container-title:Journal of Steroid Biochemistry

Author:

Kaspar Peter,Witzel Herbert

Publisher

Elsevier BV

Subject

Endocrinology,Biochemistry

Reference22 articles.

1. Steroid binding to the cytosolic estrogen receptor from rat uterus. Influence of the orientation of substituents in the 17-position of the 8β-and 8α-series;Kaspar;J. steroid Biochem.,1985

2. Chemical and biological properties of some 17-substituted estradiol derivates;Counsell;J. med. Chem.,1966

3. The preparation and pharmacology of some 3-desoxyestratrienes. Lipidshifting and estrogenic effects;Goldkamp;J. med. Chem.,1965

4. Struktur-Stoffwechsel-Wirkungsbezie-hungen bei 17α-CH2X-substituierten Östra-1,3,5(10)-trienen;Hörhold;Pharmazie,1975

5. Structural information from OH stretching frequencies. Monohydric saturated alcohols;van der Maas;Spectr. Acta,1974

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