Improvement in glucocorticoid receptor binding affinity concomitant to shift from antagonist to agonist activity in a series of 17β-carboxamide derivatives of dexamethasone-Reference-Cited by-同舟云学术

Improvement in glucocorticoid receptor binding affinity concomitant to shift from antagonist to agonist activity in a series of 17β-carboxamide derivatives of dexamethasone

Published:1989-10 Issue:4 Volume:33 Page:557-563
ISSN:0022-4731
Container-title:Journal of Steroid Biochemistry
language:en
Short-container-title:Journal of Steroid Biochemistry

Author:

Lefebvre Philippe,Formstecher Pierre,Rousseau Guy G.,Lustenberger P.,Dautrevaux Michel

Publisher

Elsevier BV

Subject

Endocrinology,Biochemistry

Reference23 articles.

1. Development of glucocorticoid antagonists;Chrousos;Pharmac. Ther.,1983

2. Unique long acting antiglucocorticoid in whole and in broken cell system;Simons,1980

3. Glucocorticoid versus anti-glucocorticoid activity: can a single functional group modification always convey antiglucocorticoid activity;Lamontagne;Endocrinology,1984

4. Glucocorticoid agonist and antagonist activity of 17–21 acetonide derivatives;Rousseau;J. steroid Biochem.,1983

5. Synthesis of steroidal 17β-carboxamide derivatives;Formstecher;Steroids,1980

Cited by 6 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Estimation of lipophilicity and design of new 17β-carboxamide glucocorticoids using RP-HPLC and quantitative structure-retention relationships analysis;Acta Chromatographica;2021-09-07

2. Evaluation of Biological Activity and Computer-Aided Design of New Soft Glucocorticoids;Archiv der Pharmazie;2017-04-18

3. Dissociated non-steroidal glucocorticoids: tuning out untoward effects;Expert Opinion on Therapeutic Patents;2007-01

4. Higher levels of control: modulation of steroid hormone-regulated gene transcription;Molecular Endocrinology;1992-07-01

5. Aldosterone antagonists destabilize the mineralocorticosteroid receptor;Biochemical Journal;1992-03-15