The affinity alkylators, 11α-bromoacetoxyprogesterone and estrone 3-bromoacetate, modify a common histidyl residue in the active site of human placental 17β,20α-hydroxysteroid dehydrogenase-Reference-Cited by-同舟云学术

The affinity alkylators, 11α-bromoacetoxyprogesterone and estrone 3-bromoacetate, modify a common histidyl residue in the active site of human placental 17β,20α-hydroxysteroid dehydrogenase

Published:1986-07 Issue:1 Volume:25 Page:103-108
ISSN:0022-4731
Container-title:Journal of Steroid Biochemistry
language:en
Short-container-title:Journal of Steroid Biochemistry

Author:

Thomas James L.,Asibey-Berko Ebenezer,Strickler Ronald C.

Publisher

Elsevier BV

Subject

Endocrinology,Biochemistry

Reference18 articles.

1. 20α-Hydroxy-steroid dehydrogenase activity a function of human placental 17β-hydroxysteroid dehydrogenase;Purdy;Biochim. biophys. Acta,1964

2. Estradiol 17β-dehydro-genase and 20α-hydroxy steroid dehydrogenase from human placental cytosol: One enzyme with two activities?;Strickler;Steroids,1980

3. 20α-Hydroxysteroid dehydrogenase and 17β-estradiol dehydrogenase localise in the cytosol of human term placenta;Strickler;Am. J. Physiol.,1982

4. Human placental 17β-estradiol dehydrogenase and 20α-hydroxysteroid dehydrogenase: Two activities at a single enzyme active site;Strickler;J. biol. Chem.,1981

5. Human placental 17β-estradiol dehydrogenase and 20α-hydroxysteroid dehydrogenase: Studies with 6β-bromoacetoxyprogesterone;Thomas;J. biol. Chem.,1983

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2. Inhibitors of 17β-Hydroxysteroid Dehydrogenases;Current Medicinal Chemistry;2003-03-01

3. A concerted, rational design of type 1 17β‐hydroxysteroid dehydrogenase inhibitors: estradiol‐adenosine hybrids with high affinity;The FASEB Journal;2002-09-05

4. Overview of a rational approach to design type I 17β-hydroxysteroid dehydrogenase inhibitors without estrogenic activity: chemical synthesis and biological evaluation;The Journal of Steroid Biochemistry and Molecular Biology;1998-08

5. A 6β-(thiaheptanamide) derivative of estradiol as inhibitor of 17β-hydroxysteroid dehydrogenase type 1;The Journal of Steroid Biochemistry and Molecular Biology;1998-02