Author:
Perno Carlo-Federico,Santoro Nadia,Balestra Emanuela,Aquaro Stefano,Cenci Alessandra,Lazzarino Giuseppe,Di Pierro Donato,Tavazzi Barbara,Balzarini Jan,Garaci Enrico,Grimaldi Settimio,Caliò Raffaele
Reference44 articles.
1. Balzarini, J. and De Clercq, E. (1991) 5-Phosphoribosyl-1-pyrophosphate synthetase converts the acyclic nucleoside phosphonates 9-(3-hydroxy-2-phosphonylmethoxypropyl)adenine and 9-(2-phosphonylmethoxyethyl)adenine directly to their antivirally active diphosphate derivatives. J. Biol. Chem. 266, 8686–8689.
2. Balzarini, J., Naesens, L., Herdewijn, P., Rosenberg, I., Holy, A., Pauwels, R., Baba, M., Johns, D.G. and De Clercq, E. (1989) Marked in vivo antiretrovirus activity of 9-(2-phosphonylmethoxyethyl)adenine, a selective anti-human immunodeficiency virus agent. Proc. Natl. Acad. Sci. USA 86, 332–336.
3. Balzarini, J., Perno, C.F., Schols, D. and De Clercq, E. (1991a) Activity of acyclic nucleoside phosphonates analogues against human immunodeficiency virus in monocyte/macrophages and peripheral blood lymphocytes. Biochem. Biophys. Res. Commun. 178, 329–335.
4. Balzarini, J., Hao, Z., Herdewijn, P., Johns, D.G. and De Clercq, E. (1991b) Intracellular metabolism and mechanism of anti-retrovirus action of 9-(2-phosphonylmethoxyethyl)adenine, a potent anti-human immunodeficiency virus compound. Proc. Natl. Acad. Sci. USA 88, 1499–1503.
5. Barditch-Crovo, P.A., Toole, J., Burgee, H., Wachsman, M., Ebeling, D., Cundy, K.C. and Jaffe H.S. (1995) A randomized, double-blind, placebo-controlled phase I/II evaluation of 9-[2-(bispivaloyloxy-methyl)phosphonyl-methoxy]adenine (Bis-POM PMEA), an orally bioavailable prodrug of the anti-HIV nucleotide, PMEA. Antiviral Res. 26, A229.
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