Antimalarial naphthoquinones. Synthesis via click chemistry, in vitro activity , docking to Pf DHODH and SAR of lapachol-based compounds-Reference-Cited by-同舟云学术

Antimalarial naphthoquinones. Synthesis via click chemistry, in vitro activity , docking to Pf DHODH and SAR of lapachol-based compounds

Published:2018-02 Issue: Volume:145 Page:191-205
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Brandão Geraldo Célio,Rocha Missias Franciele C.,Arantes Lucas Miquéias,Soares Luciana Ferreira,Roy Kuldeep K.,Doerksen Robert J.,Braga de Oliveira Alaide,Pereira Guilherme Rocha^ORCID

Funder

FAPEMIG – Fundação de Amparo à Pesquisa de Minas Gerais (Brazil)

CAPES - Coordenação e Aperfeiçoamento de Pessoal de Nível Superior (Brazil)

CNPq-Conselho Nacional de Desenvolvimento Científico e Tecnológico (Brazil)

PRONEX Rede Malária

FAPEMIG

CAPES

CNPq

National Institutes of Health (NIH) National Center for Research Resources

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference60 articles.

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5. Antimalarial activity of phenazines from lapachol, beta-lapachone and its derivatives against Plasmodium falciparum in vitro and Plasmodium berghei in vivo;de Andrade-Neto;Bioorg. Med. Chem. Lett,2004

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