Discovery of novel bromophenol 3,4-dibromo-5-(2-bromo-3,4-dihydroxy-6-(isobutoxymethyl)benzyl)benzene-1,2-diol as protein tyrosine phosphatase 1B inhibitor and its anti-diabetic properties in C57BL/KsJ-db/db mice-Reference-Cited by-同舟云学术

Discovery of novel bromophenol 3,4-dibromo-5-(2-bromo-3,4-dihydroxy-6-(isobutoxymethyl)benzyl)benzene-1,2-diol as protein tyrosine phosphatase 1B inhibitor and its anti-diabetic properties in C57BL/KsJ-db/db mice

Published:2013-06 Issue: Volume:64 Page:129-136
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Jiang Bo,Guo Shuju,Shi Dayong,Guo Chao,Wang Tao

Funder

National Natural Science Foundation of China

Natural Science Foundation of Jiangsu Province

Nantong Municipal Natural Science Foundation

Qingdao Municipal Natural Science Foundation

Shangdong Excellent Young Scientists Award Fund

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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3. Management of type 2 diabetes: new and future developments in treatment;Tahrani;Lancet,2011

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1. Recent updates on development of protein-tyrosine phosphatase 1B inhibitors for treatment of diabetes, obesity and related disorders;Bioorganic Chemistry;2022-04

2. Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic properties;Bioorganic Chemistry;2021-03

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4. Antidiabetic activity in vitro and in vivo of BDB, a selective inhibitor of protein tyrosine phosphatase 1B, from Rhodomela confervoides;British Journal of Pharmacology;2020-08-30

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