Continued exploration of 1,2,4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX isoform that selectively kill cancer cells in hypoxic environment-Reference-Cited by-同舟云学术

Continued exploration of 1,2,4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX isoform that selectively kill cancer cells in hypoxic environment

Published:2019-02 Issue: Volume:164 Page:92-105
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Krasavin Mikhail^ORCID,Shetnev Anton^ORCID,Sharonova Tatyana,Baykov Sergey^ORCID,Kalinin Stanislav,Nocentini Alessio^ORCID,Sharoyko Vladimir,Poli Giulio,Tuccinardi Tiziano^ORCID,Presnukhina Sofia,Tennikova Tatiana B.^ORCID,Supuran Claudiu T.^ORCID

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference52 articles.

1. Structure and function of carbonic anhydrases;Supuran;Biochem. J.,2016

2. Multiple binding modes of inhibitors to carbonic anhydrases: how to design specific drugs targeting 15 different isoforms?;Alterio;Chem. Rev.,2012

3. Carbonic anhydrase inhibitors and activators for novel therapeutic applications;Supuran;Future Med. Chem.,2011

4. The η-class carbonic anhydrases as drug targets for antimalarial agents;Supuran;Expert Opin. Ther. Targets,2015

5. Diuretics: from classical carbonic anhydrase inhibitors to novel applications of the sulfonamides;Supuran;Curr. Pharmaceut. Des.,2008

Cited by 58 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Unveiling the Anti-cancer Potential of Oxadiazole Derivatives: A Comprehensive Exploration of Structure-Activity Relationships and Chemico-Biological Insights;Medicinal Chemistry;2024-08-29

2. In‐vitro and in‐silico investigations of SLC‐0111 hydrazinyl analogs as human carbonic anhydrase I, II, IX, and XII inhibitors;Archiv der Pharmazie;2024-05-07

3. Chemistry of heterocycles as carbonic anhydrase inhibitors: A pathway to novel research in medicinal chemistry review;Archiv der Pharmazie;2024-04-29

4. Benzocaine-N-acylindoline conjugates: synthesis and antiviral activity against Coxsackievirus B3;Medicinal Chemistry Research;2024-02-13

5. Carbonic Anhydrase Inhibitors Induce Ferroptosis through Inhibition of AKT/FTH1 Signaling in Ewing Sarcoma Tumor Cells;Cancers;2023-10-31