Design and synthesis of novel 3-amino-5-phenylpyrazole derivatives as tubulin polymerization inhibitors targeting the colchicine-binding site

Author:

Yang Yang,Cao Yan,Yu Jingwen,Yu Xinyu,Guo Yali,Wang Fei,Ren Qingjia,Li Caolong

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference49 articles.

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3. Review: tubulin function, action of antitubulin drugs, and new drug development;Pellegrini;Cancer Invest.,2005

4. An emerging role for tubulin isotypes in modulating cancer biology and chemotherapy resistance;Parker;Int. J. Mol. Sci.,2017

5. Microtubule associated proteins as targets for anticancer drug development;Ska;Bioorg. Chem.,2021

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