Design, synthesis, and biological evaluation of first-in-class indomethacin-based PROTACs degrading SARS-CoV-2 main protease and with broad-spectrum antiviral activity-Reference-Cited by-同舟云学术

登录注册会员服务联系我们

Design, synthesis, and biological evaluation of first-in-class indomethacin-based PROTACs degrading SARS-CoV-2 main protease and with broad-spectrum antiviral activity

Published:2024-03 Issue: Volume:268 Page:116202
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Desantis Jenny,Bazzacco Alessandro,Eleuteri Michela,Tuci Sara,Bianconi Elisa,Macchiarulo Antonio,Mercorelli Beatrice,Loregian Arianna,Goracci Laura^ORCID

Funder

University of Padua

Airc Italian Foundation for Cancer Research

Ministero dell'Istruzione dell'Universita e della Ricerca

Fondazione Cassa di Risparmio di Padova e Rovigo

European Union

Publisher

Elsevier BV

Reference102 articles.

1. The PROTAC gold rush;Garber;Nat. Biotechnol.,2022

2. Major advances in targeted protein degradation: PROTACs, LYTACs, and MADTACs;Alabi;J. Biol. Chem.,2021

3. PROTACs: great opportunities for academia and industry (an update from 2020 to 2021);He;Signal Transduct. Targeted Ther.,2022

4. PROTACS: a technology with a gold rush-like atmosphere;Wang;Eur. J. Med. Chem.,2023

5. A bibliometric analysis of PROTAC from 2001 to 2021;Li;Eur. J. Med. Chem,2022

Cited by 5 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Between Theory and Practice: Computational/Experimental Integrated Approaches to Understand the Solubility and Lipophilicity of PROTACs;Journal of Medicinal Chemistry;2024-09-13

2. Human E3 ubiquitin ligases: accelerators and brakes for SARS-CoV-2 infection;Biochemical Society Transactions;2024-09-02

3. E3 ubiquitin ligase FBXO22 inhibits SARS‐CoV‐2 replication via promoting proteasome‐dependent degradation of NSP5;Journal of Medical Virology;2024-09

4. Application and challenges of nitrogen heterocycles in PROTAC linker;European Journal of Medicinal Chemistry;2024-07

5. Use of ionic liquids in amidation reactions for proteolysis targeting chimera synthesis;Organic & Biomolecular Chemistry;2024

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号京ICP备18003416号-3