A chemical modification of a peroxisome proliferator-activated receptor pan agonist produced a shift to a new dual alpha/gamma partial agonist endowed with mitochondrial pyruvate carrier inhibition and antidiabetic properties
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Published:2024-09
Issue:
Volume:275
Page:116567
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ISSN:0223-5234
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Container-title:European Journal of Medicinal Chemistry
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language:en
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Short-container-title:European Journal of Medicinal Chemistry
Author:
Laghezza Antonio,
Cerchia Carmen,
Genovese Massimo,
Montanari Roberta,
Capelli Davide,
Wackerlig Judith,
Simic Stefan,
Falbo Emanuele,
Pecora Lucia,
Leuci Rosalba,
Brunetti Leonardo,
Piemontese Luca,
Tortorella Paolo,
Biswas Abanish,
Singh Ravi Pratap,
Tambe Suhas,
Sudeep C.A.,
Pattnaik Ashok Kumar,
Jayaprakash Venkatesan,
Paoli Paolo,
Lavecchia Antonio,
Loiodice FulvioORCID