Discovery of new piperaquine hybrid analogs linked by triazolopyrimidine and pyrazolopyrimidine scaffolds with antiplasmodial and transmission blocking activities

Author:

Feitosa Livia M.,Franca Rodolfo Rodrigo F.,Ferreira Maria de Lourdes G.,Aguiar Anna C.C.,de Souza Guilherme E.,Maluf Sarah El Chamy,de Souza Juliana O.,Zapata Luana,Duarte Denise,Morais Ines,Nogueira Fatima,Nonato M. Cristina,Pinheiro Luiz C.S.ORCID,Guido Rafael V.C.,Boechat Nubia

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference49 articles.

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4. Resistance to artemisinin combination therapies (ACTs): do not forget the partner drug;Nsanzabana;Trav. Med. Infect. Dis.,2019

5. Association of Plasmodium falciparum kelch13 R561H genotypes with delayed parasite clearance in Rwanda: an open-label, single-arm, multicentre, therapeutic efficacy study;Uwimana;Lancet Infect. Dis.,2021

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