Enhanced antimalarial activity of plasmepsin V inhibitors by modification of the P 2 position of PEXEL peptidomimetics-Reference-Cited by-同舟云学术

Enhanced antimalarial activity of plasmepsin V inhibitors by modification of the P 2 position of PEXEL peptidomimetics

Published:2018-06 Issue: Volume:154 Page:182-198
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Nguyen William,Hodder Anthony N.,de Lezongard Richard Bestel,Czabotar Peter E.,Jarman Kate E.,O'Neill Matthew T.,Thompson Jennifer K.,Jousset Sabroux Helene,Cowman Alan F.,Boddey Justin A.,Sleebs Brad E.^ORCID

Funder

National Health and Medical Research Council

CASS Foundation Science and Medicine

Australian Cancer Research Foundation

Victorian State Government Operational Infrastructure

Australian Government

Howard Hughes International Scholar

NHMRC Research Fellows

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference54 articles.

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3. Four plasmepsins are active in the Plasmodium falciparum food vacuole, including a protease with an active-site histidine;Banerjee;Proc. Natl. Acad. Sci. U.S.A.,2002

4. The role of Plasmodium falciparum food vacuole plasmepsins;Liu;J. Biol. Chem.,2005

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