Structural insight into the optimization of ethyl 5-hydroxybenzo[g]indol-3-carboxylates and their bioisosteric analogues as 5-LO/m-PGES-1 dual inhibitors able to suppress inflammation-Reference-Cited by-同舟云学术

Structural insight into the optimization of ethyl 5-hydroxybenzo[g]indol-3-carboxylates and their bioisosteric analogues as 5-LO/m-PGES-1 dual inhibitors able to suppress inflammation

Published:2018-07 Issue: Volume:155 Page:946-960
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Bruno Ferdinando,Errico Suann,Pace Simona,Nawrozkij Maxim B.,Mkrtchyan Arthur S.,Guida Francesca,Maisto Rosa,Olgaç Abdurrahman,D'Amico Michele,Maione Sabatino,De Rosa Mario,Banoglu Erden^ORCID,Werz Oliver,Fiorentino Antonio^ORCID,Filosa Rosanna^ORCID

Funder

MIUR

Russian Foundation for Basic Research

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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