Optimization of a 1,3,4-oxadiazole series for inhibition of Ca2+/calmodulin-stimulated activity of adenylyl cyclases 1 and 8 for the treatment of chronic pain-Reference-Cited by-同舟云学术

Optimization of a 1,3,4-oxadiazole series for inhibition of Ca2+/calmodulin-stimulated activity of adenylyl cyclases 1 and 8 for the treatment of chronic pain

Published:2019-01 Issue: Volume:162 Page:568-585
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Kaur Jatinder,Soto-Velasquez Monica,Ding Zhong,Ghanbarpour Ahmadreza,Lill Markus A.,van Rijn Richard M.^ORCID,Watts Val J.,Flaherty Daniel P.^ORCID

Funder

National Institutes of Health

Department of Medicinal Chemistry

Molecular Pharmacology Research Enhancement Award

Purdue College of Pharmacy

Indiana CTSI Postdoctoral Challenge

Purdue Chemical Genomics Facility

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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4. Designing safer analgesics via μ-opioid receptor pathways;Chan;Trends Pharmacol. Sci.,2017

5. Isoforms of mammalian adenylyl cyclase: multiplicities of signaling;Sunahara;Mol. Interv.,2002

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