Discovery and preliminary evaluation of 2-aminobenzamide and hydroxamate derivatives containing 1,2,4-oxadiazole moiety as potent histone deacetylase inhibitors-Reference-Cited by-同舟云学术

Discovery and preliminary evaluation of 2-aminobenzamide and hydroxamate derivatives containing 1,2,4-oxadiazole moiety as potent histone deacetylase inhibitors

Published:2015-05 Issue: Volume:96 Page:1-13
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Cai Jin,Wei Hongtao,Hong Kwon Ho,Wu Xiaoqing,Cao Meng,Zong Xi,Li Lushen,Sun Chunlong,Chen Junqing,Ji Min

Funder

The Fundamental Research Funds for the Central Universities

Technology Supporting Program of Jiangsu province

National Basin Research Program of China

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference50 articles.

1. The Rpd3/Hda1 family of lysine deacetylases: from bacteria and yeast to mice and men;Yang;Nat. Rev. Mol. Cell. Biol.,2008

2. Histone lysine demethylases and their impact on epigenetics;Trojer;Cell,2006

3. Chromatin modifications and their function;Kouzarides;Cell,2007

4. Further insights into the SAR of alpha-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A;Pieroni;Eur. J. Med. Chem.,2015

5. Histone acetyltransferases;Roth;Annu. Rev. Biochem.,2001

Cited by 47 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Heterocycles–Containing HDAC Inhibitors Active in Cancer: An Overview of the Last Fifteen Years;ChemMedChem;2024-08-29

2. Preparation of Novel 3,4,5‐Triaryl‐1,2,4‐Oxadiazole Derivatives: Molecular Docking and α‐Glucosidase assessment;ChemistrySelect;2024-02-06

3. Design, Synthesis and Anti-fungal Activity of 1,2,4-Oxadiazole Derivatives Containing Diamide Moiety;CHEM J CHINESE U;2023

4. Synthesis and cytotoxic activity of N-[(alkylsulfanyl)methyl]- and N-[(arylsulfanyl)methyl]benzamides;Russian Chemical Bulletin;2023-10

5. Significance of Five-Membered Heterocycles in Human Histone Deacetylase Inhibitors;Molecules;2023-07-27