Cu (I) catalyzed alkyne-azide 1,3-dipolar cycloaddition (CuAAC): Synthesis of 17α-[1-(substituted phenyl)-1,2,3-triazol-4-yl]-19-nor-testosterone-17β-yl acetates targeting progestational and antipro-liferative activities-Reference-Cited by-同舟云学术

Cu (I) catalyzed alkyne-azide 1,3-dipolar cycloaddition (CuAAC): Synthesis of 17α-[1-(substituted phenyl)-1,2,3-triazol-4-yl]-19-nor-testosterone-17β-yl acetates targeting progestational and antipro-liferative activities

Published:2015-06 Issue: Volume:97 Page:75-82
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Mohamed Z.H.,El-Koussi Nawal A.,Mahfouz Nadia M.,Youssef Adel F.,Abdel Jaleel Gehad A.,Shouman Samia A.

Funder

The National Cancer Institute (NCI)

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference32 articles.

1. Synthesis of D-ring-substituted (5′R)- and (5′S)-17β-pyrazolinylandrostene epimers and comparison of their potential anticancer activities

2. Conformational adaptation of nuclear receptor ligand binding domains to agonists: Potential for novel approaches to ligand design

3. Progesterone Receptor Ligand Binding Pocket Flexibility: Crystal Structures of the Norethindrone and Mometasone Furoate Complexes

4. Click Chemistry: 1,2,3-Triazoles as Pharmacophores

5. Rapid Synthesis of Triazole-Modified Resveratrol Analogues via Click Chemistry

Cited by 14 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Synthetic Transformations of Higher Terpenoids. 44#. Synthesis of New Derivatives of 18-Nor-4-Amino-8(17),13,14-Labdatriene and Evaluation of Their Cytotoxicity for MCF7, HepG2, and HeLa Tumor Cell Lines;Chemistry of Natural Compounds;2024-03

2. Steroid-triazole conjugates: A brief overview of synthesis and their application as anticancer agents;Steroids;2023-09

3. Facile, Single‐Step Synthesis of a Series of D‐Ring Ethisterones Substituted with 1,4‐1,2,3‐Triazoles: Preliminary Evaluation of Cytotoxic Activities;ChemMedChem;2023-03-22

4. Synthesis of 1,2,3-Triazolyl-Substituted Derivatives of the Alkaloids Sinomenine and Tetrahydrothebaine on Ring A and Their Analgesic Activity;Chemistry of Natural Compounds;2022-09

5. Recyclable and reusable ionic liquid-supported azo precursors in Mitsunobu reactions;Organic & Biomolecular Chemistry;2022