Experience-based discovery (EBD) of aryl hydrazines as new scaffolds for the development of LSD1/KDM1A inhibitors-Reference-Cited by-同舟云学术

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Experience-based discovery (EBD) of aryl hydrazines as new scaffolds for the development of LSD1/KDM1A inhibitors

Published:2019-03 Issue: Volume:166 Page:432-444
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Li Zhong-Rui,Wang Shuai,Yang Linlin,Yuan Xiao-Han,Suo Feng-Zhi,Yu Bin^ORCID,Liu Hong-Min^ORCID

Funder

National Natural Science Foundation of China

state key laboratory of Pharmaceutical Biotechnology, Nan-jing University, China

Scientific Program of Henan Province

China Postdoctoral Science Foundation

Key Research Program of Higher Education of Henan Province

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference70 articles.

1. Histone demethylases and their roles in cancer epigenetics;D'Oto;Journal of Medical Oncology and Therapeutics,2016

2. LSD1 demethylates histone and non-histone proteins;Nicholson;Epigenetics,2009

3. Structural basis for KDM5A histone lysine demethylase inhibition by diverse compounds;Horton John;Cell Chemical Biology,2016

4. Histone lysine demethylases: emerging roles in development, physiology and disease;Shi;Nat. Rev. Genet.,2007

5. Selective inhibition of lysine-specific demethylase 5A (KDM5A) using a rhodium(III) complex for triple-negative breast cancer therapy;Yang;Angew. Chem. Int. Ed.,2018

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