Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors-Reference-Cited by-同舟云学术

Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors

Published:2016-01 Issue: Volume:108 Page:701-719
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Baltus Christine B.,Jorda Radek,Marot Christophe,Berka Karel^ORCID,Bazgier Václav,Kryštof Vladimír,Prié Gildas,Viaud-Massuard Marie-Claude

Funder

Labex

Medical Research Fondation (FRM

Ministry of Education, Youth and Sports of the Czech Republic

Czech Science Foundation

Palacky University in Olomouc

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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4. Cyclins and Cdks in development and cancer: a perspective;Deshpande;Oncogene,2005

5. Emerging drug profile: cyclin-dependent kinase inhibitors;Blachly;Leukemia Lymphoma,2013

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