Michael acceptor approach to the design of new salvinorin A-based high affinity ligands for the kappa-opioid receptor-Reference-Cited by-同舟云学术

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Michael acceptor approach to the design of new salvinorin A-based high affinity ligands for the kappa-opioid receptor

Published:2014-10 Issue: Volume:85 Page:818-829
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Polepally Prabhakar R.,Huben Krzysztof,Vardy Eyal,Setola Vincent,Mosier Philip D.,Roth Bryan L.,Zjawiony Jordan K.

Funder

NIH

University of North Carolina Chapel Hill

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference30 articles.

1. Salvinorin, a new trans-neoclerodane diterpene from Salvia divinorum (Labiatae);Ortega;J. Chem. Soc. Perkins Trans. 1,1982

2. Salvinorin A: a potent naturally occurring nonnitrogenous κ opioid selective agonist;Roth;Proc. Natl. Acad. Sci. U. S. A.,2002

3. Neuropharmacology of the naturally occurring κ-opioid hallucinogen salvinorin A;Cunningham;Pharmacol. Rev.,2011

4. Synthesis and biological evaluation of new salvinorin A analogues incorporating natural amino acids;Fichna;Bioorg. Med. Chem. Lett.,2011

5. Synthesis of neoclerodane diterpenes and their pharmacological effects;Lovell;Top. Curr. Chem.,2011

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1. Discovery of Novel, Selective, and Nonbasic Agonists for the Kappa-Opioid Receptor Determined by Salvinorin A-Based Virtual Screening;Journal of Medicinal Chemistry;2024-08-01

2. From Plant to Chemistry: Sources of Active Opioid Antinociceptive Principles for Medicinal Chemistry and Drug Design;Molecules;2023-10-14

3. Heteroaromatic salvinorin A analogue (P-3 l) elicits antinociceptive and anxiolytic-like effects;Fitoterapia;2023-06

4. Solving an Old Puzzle: Elucidation and Evaluation of the Binding Mode of Salvinorin A at the Kappa Opioid Receptor;Molecules;2023-01-11

5. Critical interactions between opioid and cannabinoid receptors during tolerance and physical dependence development to opioids in the murine gastrointestinal tract: proof of concept;Pharmacological Reports;2021-06-16

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