Discovery of a potent MLL1 and WDR5 protein-protein interaction inhibitor with in vivo antitumor activity
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
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1. Ribosome subunit attrition and activation of the p53-MDM4 axis dominate the response of MLL-rearranged cancer cells to WDR5 WIN site inhibition;ELIFE;2024
2. Ribosome subunit attrition and activation of the p53–MDM4 axis dominate the response of MLL-rearranged cancer cells to WDR5 WIN site inhibition;eLife;2024-04-29
3. Ribosome subunit attrition and activation of the p53–MDM4 axis dominate the response of MLL-rearranged cancer cells to WDR5 WIN site inhibition;2024-04-10
4. Chemical inhibitors targeting histone methylation readers;Pharmacology & Therapeutics;2024-04
5. WD Repeat Domain 5 Inhibitors for Cancer Therapy: Not What You Think;Journal of Clinical Medicine;2024-01-03
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