Design, synthesis and in vitro evaluation of novel SARS-CoV-2 3CLpro covalent inhibitors-Reference-Cited by-同舟云学术

Design, synthesis and in vitro evaluation of novel SARS-CoV-2 3CLpro covalent inhibitors

Published:2022-02 Issue: Volume:229 Page:114046
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Stille Julia K.^ORCID,Tjutrins Jevgenijs,Wang Guanyu^ORCID,Venegas Felipe A.,Hennecker Christopher^ORCID,Rueda Andrés M.,Sharon Itai,Blaine Nicole,Miron Caitlin E.,Pinus Sharon^ORCID,Labarre Anne^ORCID,Plescia Jessica^ORCID,Burai Patrascu Mihai^ORCID,Zhang Xiaocong,Wahba Alexander S.,Vlaho Danielle^ORCID,Huot Mitchell J.,Schmeing T. Martin^ORCID,Mittermaier Anthony K.,Moitessier Nicolas^ORCID

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference76 articles.

1. SARS-CoV-2 in fruit bats, ferrets, pigs, and chickens: an experimental transmission study;Schlottau;Lancet Micr,2020

2. A review of studies on animal reservoirs of the SARS coronavirus;Shi;Virus Res.,2008

3. Temporal estimates of case-fatality rate for COVID-19 outbreaks in Canada and the United States;Abdollahi;Can. Med. Assoc. J.,2020

4. WHO Coronavirus Disease;Organization,2020

5. Estimating COVID-19 mortality in Italy early in the COVID-19 pandemic;Modi;Nat. Commun.,2021

Cited by 49 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Covalent small-molecule inhibitors of SARS-CoV-2 Mpro: Insights into their design, classification, biological activity, and binding interactions;European Journal of Medicinal Chemistry;2024-11

2. Structural Basis of Main Proteases of Coronavirus Bound to Bofutrelvir;Journal of Molecular Biology;2024-11

3. How many organic small molecules might be used to treat COVID-19? From natural products to synthetic agents;European Journal of Medicinal Chemistry;2024-11

4. Crystal structures of coronaviral main proteases in complex with the non-covalent inhibitor X77;International Journal of Biological Macromolecules;2024-09

5. MOLECULAR MODELLING AND THEORETICAL DESIGN OF NOVEL NIRMATRELVIR DERIVATIVES AS SARS-COV-2 ENTRY INHIBITORS;New Materials, Compounds and Applications;2024-08-08