Synthesis, structure-activity relationships and molecular docking studies of phenyldiazenyl sulfonamides as aromatase inhibitors

Author:

Giampietro LetiziaORCID,Gallorini MarialuciaORCID,Gambacorta Nicola,Ammazzalorso AlessandraORCID,De Filippis Barbara,Della Valle Alice,Fantacuzzi MarialuigiaORCID,Maccallini CristinaORCID,Mollica Adriano,Cataldi AmeliaORCID,Nicolotti Orazio,Amoroso RosaORCID

Funder

MIUR

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference57 articles.

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2. Recent progress in the discovery of next generation inhibitors of aromatase from the structure-function perspective;Ghosh;J. Med. Chem.,2016

3. Aromatase inhibitors in the treatment of breast cancer;Brueggemeier;Endocr. Rev.,2005

4. Core glycosylation of cytochrome P-450(arom). Evidence for localization of N terminus of microsomal cytochrome P-450 in the lumen;Shimozawa;J. Biol. Chem.,1993

5. Ligand- and Structure-Based Drug Design of Non-steroidal Aromatase Inhibitors (NSAIs) in Breast Cancer;Jha,2015

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