Further hit optimization of 6-(trifluoromethyl)pyrimidin-2-amine based TLR8 modulators: Synthesis, biological evaluation and structure–activity relationships-Reference-Cited by-同舟云学术

Further hit optimization of 6-(trifluoromethyl)pyrimidin-2-amine based TLR8 modulators: Synthesis, biological evaluation and structure–activity relationships

Published:2021-12 Issue: Volume:225 Page:113809
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Dolšak Ana,Šribar Dora,Scheffler Alexander^ORCID,Grabowski Maria,Švajger Urban,Gobec Stanislav,Holze Janine,Weindl Günther,Wolber Gerhard^ORCID,Sova Matej

Funder

Javna Agencija za Raziskovalno Dejavnost RS

Deutscher Akademischer Austauschdienst

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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1. Label-free biosensor assay decodes the dynamics of Toll-like receptor signaling;2024-01-20

2. Synthesis, bioactivity and preliminary mechanism of action of novel trifluoromethyl pyrimidine derivatives;Arabian Journal of Chemistry;2022-09