Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGF/p75-Reference-Cited by-同舟云学术

Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGF/p75

Published:2015-08 Issue: Volume:101 Page:288-294
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Cuzzucoli Crucitti Giuliana,Pescatori Luca,Messore Antonella,Madia Valentina Noemi,Pupo Giovanni,Saccoliti Francesco,Scipione Luigi,Tortorella Silvano,Di Leva Francesco Saverio,Cosconati Sandro,Novellino Ettore,Debyser Zeger,Christ Frauke,Costi Roberta,Di Santo Roberto

Funder

MIUR

PRIN 2010-2011

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference37 articles.

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4. Discovery of raltegravir, a potent, selective orally bioavailable HIV-integrase inhibitor for the treatment of HIV-AIDS infection;Summa;J. Med. Chem.,2008

5. Broad antiretroviral activity and resistance profile of the novel human immunodeficiency virus integrase inhibitor elvitegravir (JTK-303/GS-9137);Shimura;J. Virol.,2008

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