Synthesis and biological evaluation of a new series of 2-amino-3-aroyl thiophene derivatives as agonist allosteric modulators of the A 1 adenosine receptor. A position-dependent effect study-Reference-Cited by-同舟云学术

Synthesis and biological evaluation of a new series of 2-amino-3-aroyl thiophene derivatives as agonist allosteric modulators of the A 1 adenosine receptor. A position-dependent effect study

Published:2015-08 Issue: Volume:101 Page:185-204
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Romagnoli Romeo,Baraldi Pier Giovanni,Lopez-Cara Carlota,Cruz-Lopez Olga,Moorman Allan R.,Massink Arnault,IJzerman Adriaan P.,Vincenzi Fabrizio,Borea Pier Andrea,Varani Katia

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference66 articles.

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5. ADENOSINE REGULATES VIA TWO DIFFERENT TYPES OF RECEPTORS, THE ACCUMULATION OF CYCLIC AMP IN CULTURED BRAIN CELLS

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