Probing the ‘bipolar’ nature of the carbonic anhydrase active site: Aromatic sulfonamides containing 1,3-oxazol-5-yl moiety as picomolar inhibitors of cytosolic CA I and CA II isoforms-Reference-Cited by-同舟云学术

Probing the ‘bipolar’ nature of the carbonic anhydrase active site: Aromatic sulfonamides containing 1,3-oxazol-5-yl moiety as picomolar inhibitors of cytosolic CA I and CA II isoforms

Published:2015-08 Issue: Volume:101 Page:334-347
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Krasavin Mikhail,Korsakov Mikhail,Dorogov Mikhail,Tuccinardi Tiziano,Dedeoglu Nurcan,Supuran Claudiu T.

Funder

Russian Scientific Fund

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference37 articles.

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3. Carbonic anhydrsases: novel therapeutic applications for inhibitors and activators;Supuran;Nat. Rev. Drug Discov.,2008

4. Carbonic anhydrases: from biomedical applications of the inhibitors and activators to biotechnologic use for CO2 capture;Supuran;J. Enzyme Inhib. Med. Chem.,2013

5. New zinc binding motifs in the design of selective carbonic anhydrase inhibitors;Winum;Mini Rev. Med. Chem.,2006

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