Design, synthesis and biological evaluation of 4-anilinoquinazoline derivatives as new c-myc G-quadruplex ligands

Author:

Jiang Yin,Chen Ai-Chun,Kuang Guo-Tao,Wang Shi-Ke,Ou Tian-Miao,Tan Jia-Heng,Li Ding,Huang Zhi-Shu

Funder

Natural Science Foundation of China

Guangdong Provincial Key Laboratory of Construction Foundation

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference35 articles.

1. Quadruplex DNA: sequence, topology and structure;Burge;Nucleic Acids Res.,2006

2. G-quadruplexes and their regulatory roles in biology;Rhodes;Nucleic Acids Res.,2015

3. G-quadruplexes in RNA biology, Wiley interdisciplinary reviews;Millevoi;RNA,2012

4. Quantitative visualization of DNA G-quadruplex structures in human cells;Biffi;Nat. Chem.,2013

5. DNA secondary structures: stability and function of G-quadruplex structures;Bochman;Nat. Rev. Genet.,2012

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