Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist – Neurokinin-1 antagonist peptidomimetics
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference60 articles.
1. Opioids and their receptors: are we there yet?;Pasternak;Neuropharmacology,2014
2. Stronger antinociceptive efficacy of opioids at the injured nerve trunk than at its peripheral terminals in neuropathic pain;Labuz;J. Pharmacol. Exp. Ther.,2013
3. The loss of antinociceptive efficacy of spinal morphine in rats with nerve ligation injury is prevented by reducing spinal afferent drive;Ossipov;Neurosci. Lett.,1995
4. Cloning of a delta opioid receptor by functional expression;Evans;Science,1992
5. The delta-opioid receptor: isolation of a cDNA by expression cloning and pharmacological characterization;Kieffer;Proc. Natl. Acad. Sci. U. S. A.,1992
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