Synthesis and biological evaluations of novel endomorphin analogues containing α-hydroxy-β-phenylalanine (AHPBA) displaying mixed μ/δ opioid receptor agonist and δ opioid receptor antagonist activities-Reference-Cited by-同舟云学术

Synthesis and biological evaluations of novel endomorphin analogues containing α-hydroxy-β-phenylalanine (AHPBA) displaying mixed μ/δ opioid receptor agonist and δ opioid receptor antagonist activities

Published:2015-03 Issue: Volume:92 Page:270-281
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Hu Miao,Giulianotti Marc A.,McLaughlin Jay P.,Shao Jiaan,Debevec Ginamarie,Maida Laura E.,Geer Phaedra,Cazares Margaret,Misler Jaime,Li Ling,Dooley Colette,Ganno Michelle L.,Eans Shainnel O.,Mizrachi Elisa,Santos Radleigh G.,Yongye Austin B.,Houghten Richard A.,Yu Yongping

Funder

National Natural Science Foundation of China

Natural Science Foundation of Zhejiang Province

NIH

Arthritis & Chronic Pain Research Institute (USA)

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference77 articles.

1. Simultaneous targeting of multiple opioid receptors: a strategy to improve side-effect profile

2. Targeting opioid receptor heterodimers: Strategies for screening and drug development