Synthesis and optimization of an original V-shaped collection of 4-7-disubstituted Pyrido[3,2-d]pyrimidines as CDK5 and DYRK1A inhibitors-Reference-Cited by-同舟云学术

Synthesis and optimization of an original V-shaped collection of 4-7-disubstituted Pyrido[3,2-d]pyrimidines as CDK5 and DYRK1A inhibitors

Published:2014-06 Issue: Volume:80 Page:352-363
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Dehbi Oussama,Tikad Abdellatif,Bourg Stéphane,Bonnet Pascal,Lozach Olivier,Meijer Laurent,Aadil Mina,Akssira Mohammed,Guillaumet Gérald,Routier Sylvain

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference24 articles.

1. Protein kinases, their function and implication in cancer and other diseases;Shchemelinin;Folia Biologica (Praha),2006

2. Chemical approaches to the study of protein tyrosine kinases and their implications for mechanism and inhibitor design;Cole;Pharmacology & Therapeutics,1999

3. Cyclin-dependent kinase inhibitors: a survey of recent patent literature;Galons;Expert Opinion on Therapeutic Patents,2010

4. Cyclin-dependent kinase inhibitors closer to market launch?;Galons;Expert Opinion on Therapeutic Patents,2013

5. Synthesis of chromeno[3,4-b]indoles as Lamellarin D analogues: a novel DYRK1A inhibitor class;Neagoie;European Journal of Medicinal Chemistry,2012

Cited by 42 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. A review on synthetic inhibitors of dual-specific tyrosine phosphorylation-regulated kinase 1A (DYRK1A) for the treatment of Alzheimer’s disease (AD);Bioorganic & Medicinal Chemistry;2024-09

2. Novel Medicinal Chemistry Strategies Targeting CDK5 for Drug Discovery;Journal of Medicinal Chemistry;2023-05-26

3. Dual Specificity Tyrosine Phosphorylation-Regulated Kinase 1A (DYRK1A) Inhibitors: The Quest for a Disease-Modifying Treatment for Alzheimer’s Disease;Deciphering Drug Targets for Alzheimer’s Disease;2023

4. Characterization, biological evaluation and molecular docking of a synthesised quinazolinone-based derivative;Journal of Molecular Structure;2022-10

5. Synthesis, antimicrobial evaluation, crystal structure, Hirschfeld surface analysis and docking studies of 4-[2-(1-methyl-1H-imidazol-2-ylsulfanyl)-acetylamino]-benzenesulfonic acid;Journal of Molecular Structure;2022-10