Small molecule-induced degradation of the full length and V7 truncated variant forms of human androgen receptor-Reference-Cited by-同舟云学术

Small molecule-induced degradation of the full length and V7 truncated variant forms of human androgen receptor

Published:2018-09 Issue: Volume:157 Page:1164-1173
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Dalal Kush,Morin Helene,Ban Fuqiang,Shepherd Ashley,Fernandez Michael^ORCID,Tam Kevin J.,Li Huifang,LeBlanc Eric,Lack Nathan,Prinz Helge,Rennie Paul S.,Cherkasov Artem

Funder

Canadian Institutes of Health Research (CIHR

Prostate Cancer Canada-Translational Acceleration Grant (PCC-TAG

Terry Fox New Frontiers

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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4. Development of a second-generation antiandrogen for treatment of advanced prostate cancer;Tran;Science,2009

5. Functional analysis of androgen receptor mutations that confer anti-androgen resistance identified in circulating cell-free DNA from prostate cancer patients;Lallous;Genome Biol.,2016

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