Exploring the structure-activity relationship of benzylidene-2,3-dihydro-1H-inden-1-one compared to benzofuran-3(2H)-one derivatives as inhibitors of tau amyloid fibers-Reference-Cited by-同舟云学术

Exploring the structure-activity relationship of benzylidene-2,3-dihydro-1H-inden-1-one compared to benzofuran-3(2H)-one derivatives as inhibitors of tau amyloid fibers

Published:2022-03 Issue: Volume:231 Page:114139
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Boukherrouba Emeline,Larosa Camille^ORCID,Nguyen Kim-Anh^ORCID,Caburet Jérémy,Lunven Laurent,Bonnet Hugues^ORCID,Fortuné Antoine,Boumendjel Ahcène,Boucherle Benjamin,Chierici Sabine,Peuchmaur Marine

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference41 articles.

1. Tau in Alzheimer disease and related tauopathies;Iqbal;Curr. Alzheimer Res.,2010

2. Neuropathology of tauopathies: principles and practice;Kovacs;Neuropathol. Appl. Neurobiol.,2015

3. Tau and tauopathies;Arendt;Brain Res. Bull.,2016

4. Assembly of tau protein into Alzheimer paired helical filaments depends on a local sequence motif (306VQIVYK311) forming β structure;von Bergen;Proc. Natl. Acad. Sci. U.S.A.,2000

5. Prediction of nucleating sequences from amyloidogenic propensities of tau-related peptides;Rojas Quijano;Biochemistry,2006

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