Identification of novel indole derivatives as highly potent and efficacious LSD1 inhibitors-Reference-Cited by-同舟云学术

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Identification of novel indole derivatives as highly potent and efficacious LSD1 inhibitors

Published:2022-09 Issue: Volume:239 Page:114523
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Zhang Xiangyu,Sun Yixiang,Huang Hailan,Wang Xinran,Wu Tianxiao,Yin Wenbo,Li Xiaojia,Wang Lin,Gu Yanting,Zhao Dongmei,Cheng Maosheng

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference74 articles.

1. Histone demethylation mediated by the nuclear amine oxidase homolog LSD1;Shi;Cell,2004

2. Crystal structure of human histone lysine-specific demethylase 1 (LSD1);Chen;Proc. Natl. Acad. Sci. U.S.A.,2006

3. trans-2-Phenylcyclopropylamine is a mechanism-based inactivator of the histone demethylase LSD1;Schmidt;Biochemistry,2007

4. Structural basis for the inhibition of the LSD1 histone demethylase by the antidepressant trans-2-phenylcyclopropylamine;Yang;Biochemistry,2007

5. DNA oxidation as triggered by H3K9me2 demethylation drives estrogen-induced gene expression;Perillo;Science,2008

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3. Unveiling Arformoterol as a potent LSD1 inhibitor for breast cancer treatment: A comprehensive study integrating 3D-QSAR pharmacophore modeling, molecular docking, molecular dynamics simulations and in vitro assays;International Journal of Biological Macromolecules;2024-02

4. Lysine-Specific Demethylase 1 Inhibitors: A Comprehensive Review Utilizing Computer-Aided Drug Design Technologies;Molecules;2024-01-22

5. Sc(OTf)3-catalyzed diastereoselective [4 + 2] cycloaddition reaction of 3-benzylideneindoline-2-thiones with alkylidene malonates;Tetrahedron Letters;2024-01

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