Identification of novel chemotypes as CXCR2 antagonists via a scaffold hopping approach from a thiazolo[4,5-d]pyrimidine
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference44 articles.
1. The role of CXCR2 in acute inflammatory responses and its antagonists as anti-inflammatory therapeutics;Zhang;Curr. Opin. Hematol.,2019
2. Targeting CXCR1/2: the medicinal potential as cancer immunotherapy agents, antagonists research highlights and challenges ahead;Che;Eur. J. Med. Chem.,2020
3. Role of chemokines in tumor growth;Raman;Cancer Lett.,2007
4. Potential roles and targeted therapy of the CXCLs/CXCR2 Axis in cancer and inflammatory diseases;Cheng;Biochim. Biophys. Acta Rev. Canc,2019
5. A potent and selective nonpeptide antagonist of CXCR2 inhibits acute and chronic models of arthritis in the rabbit;Podolin;J. Immunol.,2002
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