Synthesis of 2H-Imidazo[2′,1':2,3] [1,3]thiazolo[4,5-e]isoindol-8-yl-phenylureas with promising therapeutic features for the treatment of acute myeloid leukemia (AML) with FLT3/ITD mutations

Author:

Cilibrasi Vincenzo,Spanò Virginia,Bortolozzi Roberta,Barreca Marilia,Raimondi Maria Valeria,Rocca RobertaORCID,Maruca AnnalisaORCID,Montalbano Alessandra,Alcaro Stefano,Ronca RobertoORCID,Viola GiampietroORCID,Barraja Paola

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference64 articles.

1. FLT3: ITDoes matter in leukemia;Levis;Leukemia,2003

2. The roles of FLT3 in hematopoiesis and leukemia;Gilliland;Blood,2002

3. The Surveillance, Epidemiology, and End Results (SEER) Program of the National Cancer Institute, Www.Seer.Cancer.Gov. (n.d.).

4. Receptor tyrosine kinase signalling as a target for cancer intervention strategies;Zwick;Endocr. Relat. Cancer,2001

5. Essential role of signal transducer and activator of transcription (Stat)5a but not Stat5b for Flt3-dependent signaling;Zhang;J. Exp. Med.,2000

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