Novel alpha6 preferring GABA-A receptor ligands based on loreclezole-Reference-Cited by-同舟云学术

Novel alpha6 preferring GABA-A receptor ligands based on loreclezole

Published:2022-12 Issue: Volume:244 Page:114780
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Simeone Xenia,Ernst Margot,Seidel Thomas,Heider Joerg,Enz Doris,Monticelli Serena,Vogel Florian Daniel,Koniuszewski Filip,Langer Thierry,Scholze Petra,Pace Vittorio^ORCID,Miele Margherita

Funder

Universität Wien

European Federation of Pharmaceutical Industries and Associations

Università degli Studi di Torino

European Commission

Innovative Medicines Initiative

Austrian Science Fund

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference36 articles.

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3. Structural studies of GABAA receptor binding sites: which experimental structure tells us what?;Puthenkalam;Front. Mol. Neurosci.,2016

4. Shared structural mechanisms of general anaesthetics and benzodiazepines;Kim;Nature,2020

5. α6-Containing GABAA receptors: functional roles and therapeutic potentials;Sieghart;Pharmacol. Rev.,2022

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