Pyrido[2,3-b][1,5]benzoxazepin-5(6H)-one derivatives as CDK8 inhibitors

Author:

Martínez-González Sonia,García Ana Belén,Albarrán M. Isabel,Cebriá Antonio,Amezquita-Alves Adrián,García-Campos Francisco Javier,Martínez-Gago Jaime,Martínez-Torrecuadrada Jorge,Muñoz I.G.,Blanco-Aparicio Carmen,Pastor Joaquín

Funder

H2020 Research Infrastructures

Ministerio de Economía y Competitividad

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference25 articles.

1. The mammalian mediator complex and its role in transcriptional regulation;Conaway;Trends Biochem. Sci.,2005

2. The two faces of Cdk8, a positive/negative regulator of transcription;Nemet;Biochimie,2014

3. Cyclin C is a haploinsufficient tumour suppressor;Li;Nat. Cell Biol.,2014

4. CDK8 is a colorectal cancer oncogene that regulates beta-catenin activity;Firestein;Nature,2008

5. CDK8 expression in 470 colorectal cancers in relation to beta-catenin activation, other molecular alterations and patient survival;Firestein;Int. J. Canc.,2010

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