Synthesis, biochemical, pharmacological characterization and in silico profile modelling of highly potent opioid orvinol and thevinol derivatives-Reference-Cited by-同舟云学术

Synthesis, biochemical, pharmacological characterization and in silico profile modelling of highly potent opioid orvinol and thevinol derivatives

Published:2020-04 Issue: Volume:191 Page:112145
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Szűcs Edina,Marton János,Szabó Zoltán,Hosztafi Sándor^ORCID,Kékesi Gabriella,Tuboly Gábor,Bánki László,Horváth Gyöngyi,Szabó Pál T.,Tömböly Csaba^ORCID,Varga Zsuzsanna Katalin,Benyhe Sándor^ORCID,Ötvös Ferenc

Funder

OTKA

National Research, Development and Innovation Office (NKFIH), Budapest, Hungary

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference65 articles.

1. Challenges for opioid receptor nomenclature: IUPHAR Review 9;Cox;Br. J. Pharmacol.,2015

2. Current research on opioid receptor function;Feng;Curr. Drug Targets,2012

3. Opioid receptors: from binding sites to visible molecules in vivo;Kieffer;Neuropharmacology,2009

4. Bioinformatics and evolution of vertebrate nociceptin and opioid receptors;Stewens,2015

5. Novel GPCR paradigms at the μ-opioid receptor;Thompson;Br. J. Pharmacol.,2015

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