Design, synthesis, and electrophysiological evaluation of NS6740 derivatives: Exploration of the structure-activity relationship for alpha7 nicotinic acetylcholine receptor silent activation
Author:
Funder
National Institutes of Health
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference53 articles.
1. A neuronal nicotinic acetylcholine-receptor subunit (Alpha-7) is developmentally regulated and forms a homooligomeric channel blocked by alpha-btx;Couturier;Neuron,1990
2. Molecular cloning, functional properties, and distribution of rat brain alpha7: a nicotinic cation channel highly permeable to calcium;Seguela;J. Neurosci.,1993
3. α7 Nicotinic acetylcholine receptors and their role in cognition;Lendvai;Brain Res. Bull.,2013
4. Neuronal nicotinic receptors: from structure to pathology;Gotti;Prog. Neurobiol.,2004
5. Expression and function of the cholinergic system in immune cells;Fujii;Front. Immunol.,2017
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