Design, synthesis and biological evaluation of novel O-carbamoyl ferulamide derivatives as multi-target-directed ligands for the treatment of Alzheimer’s disease

Author:

Sang Zhipei,Wang Keren,Bai Ping,Wu Anguo,Shi Jian,Liu Wenmin,Zhu Gaofeng,Wang Yiling,Lan Yu,Chen Zude,Zhao Yiyang,Qiao Zhanpin,Wang Changning,Tan Zhenghuai

Funder

TEM

China Scholarship Council

International Training of High-level Talents in Henan Province

Key Scientific Research Project of Colleges and Universities in Henan Province

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference46 articles.

1. Alzheimer’s disease;Barnett;Lancet,2019

2. World Alzheimer Report 2018—the State of the Art of Dementia Research: New Frontiers;Patterson,2018

3. Amyloid β oligomers constrict human capillaries in Alzheimer’s disease via signaling to pericytes;Nortley;Science,2019

4. Alzheimer disease: clinical use of cholinergic drugs in Alzheimer disease;Desmarais;Nat. Rev. Neurol.,2010

5. Guidelines for managing Alzheimer’s disease: Part II. Treatment;Cummings;Am. Fam. Physician,2002

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