Design and synthesis of tripeptidyl furylketones as selective inhibitors against the β5 subunit of human 20S proteasome-Reference-Cited by-同舟云学术

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Design and synthesis of tripeptidyl furylketones as selective inhibitors against the β5 subunit of human 20S proteasome

Published:2020-04 Issue: Volume:192 Page:112160
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Sun Qi,Zhou Tongliang,Xi Dandan,Li Xiaona,Lü Zirui,Xu Fengrong,Wang Chao,Niu Yan,Xu Ping

Funder

National Natural Science Foundation of China

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference31 articles.

1. Chemical and biological approaches for adapting proteostasis to ameliorate protein misfolding and aggregation diseases: progress and prognosis;Lindquist;Cold Spring Harb. Perspect. Biol.,2011

2. The ubiquitin-proteasome pathway: on protein death and cell life;Ciechanover;EMBO J.,1998

3. The 26S proteasome: a molecular machine designed for controlled proteolysis;Voges;Annu. Rev. Biochem.,1999

4. Structure of 20S proteasome from yeast at 2.4 angstrom resolution;Groll;Nature,1997

5. Subunit arrangement in the human 20S proteasome;Kopp;Proc. Natl. Acad. Sci. U.S.A.,1997

Cited by 2 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Design, synthesis, and biological evaluation of some novel naphthoquinone‐glycine/β‐alanine anilide derivatives as noncovalent proteasome inhibitors;Chemical Biology & Drug Design;2023-02-17

2. Pseudopeptides with aldehyde or vinylsulfone warheads: Synthesis and antiproteasomal activity;Bioorganic Chemistry;2021-10

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