Optimization of pyrazolo[1,5-a]pyrimidines lead to the identification of a highly selective casein kinase 2 inhibitor-Reference-Cited by-同舟云学术

Optimization of pyrazolo[1,5-a]pyrimidines lead to the identification of a highly selective casein kinase 2 inhibitor

Published:2020-12 Issue: Volume:208 Page:112770
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Krämer Andreas,Kurz Christian Georg^ORCID,Berger Benedict-Tilman^ORCID,Celik Ibrahim Ethem,Tjaden Amelie^ORCID,Greco Francesco Aleksy^ORCID,Knapp Stefan,Hanke Thomas^ORCID

Funder

SGC

AbbVie

Bayer Pharma AG

Boehringer Ingelheim, Canada Foundation for Innovation

Eshelman Institute for Innovation

Genome Canada

Innovative Medicines Initiative EUbOPEN

Janssen

Merck KGaADarmstadt Germany

MSD

Novartis Pharma AG

Ontario Ministry of Economic Development and Innovation

Pfizer

São Paulo Research Foundation- FAPESP

Takeda

Wellcome. S.K.

C.K

German cancer network

Frankfurt cancer center

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference61 articles.

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5. The ins and outs of selective kinase inhibitor development;Müller;Nat. Chem. Biol.,2015

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