Design, synthesis and biological assessment of new selective COX-2 inhibitors including methyl sulfonyl moiety
Author:
Funder
Anadolu Üniversitesi
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference44 articles.
1. Synthesis and evaluations of selective COX-2 inhibitory effects: Benzo[d]thiazol analogs
2. Structural investigation on the selective COX-2 inhibitors mediated cardiotoxicity: A review
3. COX-1/COX-2 inhibition assays and histopathological study of the new designed anti-inflammatory agent with a pyrazolopyrimidine core
4. Ligand based design and synthesis of pyrazole based derivatives as selective COX-2 inhibitors
5. Structural modification of indomethacin toward selective inhibition of COX-2 with a significant increase in van der Waals contributions
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